36-105-0R

Tocris Bioscience™ (R)-DRF053 dihydrochloride

Manufacturer: Fischer Scientific

Select a Size

Pack Size SKU Availability Price
Each of 1 36-105-0R-Each-of-1 In Stock ₹ 1,36,639.32

36-105-0R - Each of 1

₹ 1,36,639.32

In Stock

Quantity

1

Base Price: ₹ 1,36,639.32

GST (18%): ₹ 24,595.078

Total Price: ₹ 1,61,234.398

Purity

>98%

Product Type

(R)-DRF053 dihydrochloride

Inhibitors

(R)-DRF053 dihydrochloride

Quantity

50 mg

Molecular Weight (g/mol)

490.43

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Description

  • Potent casein kinase 1 (CK1) inhibitor (IC50 = 14 nM)
  • Also an ATP-competitive cyclin-dependent kinase (cdk) inhibitor (IC50 values are 0.093 - 0.29, 0.21 and 0.82 μM for cdk2, cdk5 and cdk7, respectively)
  • Shown to inhibit amyloid-β production in N2A-APP695 cells.