37-061-0R

Tocris Bioscience™ FR 180204

Manufacturer: Fischer Scientific

Select a Size

Pack Size SKU Availability Price
Each of 1 37-061-0R-Each-of-1 In Stock ₹ 30,972.72

37-061-0R - Each of 1

₹ 30,972.72

In Stock

Quantity

1

Base Price: ₹ 30,972.72

GST (18%): ₹ 5,575.09

Total Price: ₹ 36,547.81

Purity

>98%

Product Type

FR 180204

Inhibitors

FR 180204

Quantity

10 mg

Molecular Weight (g/mol)

327.34

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Description

  • Selective ERK inhibitor (IC50 values are 0.14 and 0.31 μM for ERK2 and ERK1 respectively)
  • Displays 30-fold selectivity for ERK over p38α (IC50 = 10 μM); displays no activity against human recombinant MEK1, MKK4, IKKα, PKCα, Src, Syc and PDGFα at concentrations less than 30 μM
  • Also inhibits TGFβ-induced AP-1 activation in Mv1Lu cells (IC50 = 3.1 μM).