37-261-0R

Tocris Bioscience™ GSK 429286

Manufacturer: Fischer Scientific

Select a Size

Pack Size SKU Availability Price
Each of 1 37-261-0R-Each-of-1 In Stock ₹ 37,518.06

37-261-0R - Each of 1

₹ 37,518.06

In Stock

Quantity

1

Base Price: ₹ 37,518.06

GST (18%): ₹ 6,753.251

Total Price: ₹ 44,271.311

Purity

>97%

Quantity

10 mg

Molecular Weight (g/mol)

432.37

Gene Alias

GSK429286A

Product Type

GSK 429286

Inhibitors

GSK 429286

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Description

  • Selective Rho-kinase inhibitor (IC50 values are 14, 780 and 1940 nM for ROCK1, RSK and p70S6K respectively)
  • Reverses adrenalin-induced contraction of the rat aortic ring (IC50 = 190 nM) and causes a dose-dependent decrease in mean arterial blood pressure in spontaneous hypertensive rats
  • Orally active.