50-587-60001
MilliporeSigma™ Calbiochem™ RXFP1 Agonist
Manufacturer: MilliporeSigma™
Select a Size
| Pack Size | SKU | Availability | Price |
|---|---|---|---|
| Each of 1 | 50-587-60001-Each-of-1 | In Stock | ₹ 22,416.72 |
50-587-60001 - Each of 1
In Stock
Quantity
1
Base Price: ₹ 22,416.72
GST (18%): ₹ 4,035.01
Total Price: ₹ 26,451.73
Color
White
Target Proteins
hRXFP1
Solubility
DMSO
Form
Powder
Description
98% by HPLC
Molecular Formula
C24H21F3N2O5S
Content And Storage
Protect from light
Quantity
10 mg
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Description
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- Although shown to be ∽150-fold and 500-fold less potent than relaxin (RLX), respectively, in VEGF mRNA induction and cellular impedance assays, pharmacokinetic studies reveal superior in vivo stability to RLX and in vivo bioavailability in mice via oral ( C max / T max = 604 nM/plasma/1 h and 1026 ng/g heart/1.5 h; 30mg/kg) or intraperitoneal ( C max / T max = 9.29μM/plasma/1 h and 28.6μmol/kg heart/1 h; 30mg/kg) administration with good aqueous solubility (7μM in PBS).